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Targets Recommended: PKC

30

抑制剂 & 化合物

1

TargetMol 试剂盒

2

重组蛋白

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Cat. No.	Product Name	Form	Specificity Of Inhibition
CL0112	PKC inhibitor kit PKC inhibitor kit

TargetMol 试剂盒

PKC inhibitor kit

Cat.No: CL0112

Cat. No.	Product Name	Target	Signaling Pathways
TP1955L	PKC β pseudosubstrate acetate PKC β pseudosubstrate醋酸盐,Protein kinase C beta pseudosubstrate,PKC beta pseudosubstrate,PKC β pseudosubstrate acetate (172308-76-8 Free base)	PKC	Chromatin/Epigenetic; Cytoskeletal Signaling
	PKC β pseudosubstrate acetate (PKC β pseudosubstrate acetate (172308-76-8 Free base)) 是一种选择性的、细胞渗透的 PKC 抑制剂。
T8376	PKCβ inhibitor 1 KUN79359	Apoptosis; PKC	Apoptosis; Chromatin/Epigenetic; Cytoskeletal Signaling
	PKCβ inhibitor 1 (KUN79359) 是一种 ATP 竞争性和选择性PKCβ抑制剂，对人 PKCβ1 和 PKCβ2 的IC50分别为 21 和 5 nM。
T12494	PKC-IN-1	PKC	Chromatin/Epigenetic; Cytoskeletal Signaling
	PKC-IN-1 是 ATP-竞争性可逆 PKC 抑制剂，对人 PKCβ 和 PKCα 的 Ki 值分别为 5.3 和 10.4 nM，对人 PKCα、PKCβI、PKCβII、PKCθ、PKCγ、PKC mu 和 PKCε 的IC50值分别为 2.3、8.1、7.6、25.6、57.5、314 和 808 nM。
TP1956L	PKC ζ pseudosubstrate acetate PKC ζ pseudosubstrate acetate (799764-07-1 free base)	PKC	Chromatin/Epigenetic; Cytoskeletal Signaling
	PKC ζ pseudosubstrate acetate 是蛋白激酶 C (PKC) ζ 的抑制剂；附着于细胞通透性触角足结构域载体肽。由 PKC ζ 假底物结构域的氨基酸 113-129 组成，通过二硫键连接到触角足结构域载体肽。 Antennapedia 肽在 4 或 37°C 时被完整细胞积极吸收，确保快速有效地吸收抑制肽。一旦进入细胞，二硫键在细胞质中被还原，导致抑制肽的释放。通过 PKC ζ 非依赖性途径诱导肥大细胞脱粒。
T8764	PKC-iota inhibitor 1	PKC	Chromatin/Epigenetic; Cytoskeletal Signaling
	PKC-iota inhibitor 1 是一种蛋白激酶 C-iota(PKC-ι ℩)的抑制剂，IC50值为 0.34 μM。
T35827L	PKCε Inhibitor Peptide acetate PKCε Inhibitor Peptide acetate(182683-50-7 Free base)	PKC	Chromatin/Epigenetic; Cytoskeletal Signaling
	PKCε Inhibitor Peptide acetate 是一种特异性 PKCε 抑制剂，含有其特定受体活化 C 激酶 (RACK) 的位点。 PKCε Inhibitor Peptide acetate 抑制 PKCε 的转运，但不抑制 αPKC，βPKC 和 δPKC 的转运。
T5817	PKC-theta inhibitor hcl PKC-theta inhibitor	PKC	Chromatin/Epigenetic; Cytoskeletal Signaling
	PKC-theta inhibitor hcl 是一种选择性 PKC-θ 抑制剂 (IC50:12 nM)。
T35827	Epsilon-V1-2 PKCε Inhibitor Peptide,Protein Kinase Cɛ Inhibitor Peptide,ɛV1-2
	Protein kinase C (PKC ) is a calcium-independent, phospholipid- and diacylglycerol-dependent serine/threonine kinase involved in diverse signaling pathways, including those involved in neuronal signaling, cytoskeletal function, and inflammation.[1] PKC inhibitor peptide is a synthetic peptide corresponding to an amino acid sequence found in the amino terminal C2 domain of most mammalian forms of PKC .[2] It selectively and reversibly inhibits the translocation of PKC to intracellular membrane...
T35826	PKC fragment (530-558)
	PKC fragment (530-558) 是蛋白激酶C (PKC) 的肽片段，是一种有效的 PKC 激活剂。Protein Kinase C (530-558) 可显著抑制破骨细胞骨吸收。
T80071	PKCζ/ι pseudosubstrate inhibitor
	PKCζ/ι偽基質抑制劑對PKC酶家族表現廣譜抑制作用，並可能促成記憶功能障礙。
T75885	PKC β pseudosubstrate TFA
	PKCβ pseudosubstrate TFA 是一种选择性的、细胞渗透的 PKC 抑制剂。
T76412	PKCδ Peptide Substrate
	PKCδPeptide Substrate 是一种δ-typePKC 的特异性底物，其序列与含有 Thr-431 的小鼠 eEF-1α 序列 422-443 相对应。
T61604	PKC-IN-4
	PKC-IN-4 (compound 7l) is a highly potent and orally active inhibitor of atypical protein kinase C (aPKC), exhibiting an IC 50 value of 0.52 μM. In vitro studies have demonstrated that PKC-IN-4 effectively suppresses NF-κB activity induced by TNF-α. Moreover, this compound effectively impedes the permeability of the retinal vasculature, induced by both VEGF and TNFα. [1]
T71993	PKC-9
	PKC-9 is a PKC-zeta inhibitor 9.
T83754	PKCδ Substrate TFA Protein Kinase Cδ Substrate
	PKCδ substrate是一种用于PKCδ的肽基底，常用于无细胞及细胞内测定中监测PKCδ活性。
T80248	PKCε (85-92)	PKC	Chromatin/Epigenetic; Cytoskeletal Signaling
	PKCε(85-92) 是一种具有生物活性的肽，其作为 e-PKC 特异性激活剂，能够促进野生型细胞中的 MARCKS 磷酸化作用，对基因敲除小鼠来源的细胞中的 MARCKS 磷酸化则无影响。
T62945	Aurora A/PKC-IN-1
	Aurora A/PKC-IN-1 (Compound 2e) 是一种有效的 Aurora A (AurA) 和 PKC (α, β1, β2, θ) 双重抑制剂，作用于 AurA (IC50: 6.9 nM) 和 PKCα (IC50: 16.9 nM)。Aurora A/PKC-IN-1 对乳腺癌细胞表现出抗增殖和抗转移作用。
T80511	PKCε inhibitor peptide,myristoylated Myr‐PKCɛ-	PKC	Chromatin/Epigenetic; Cytoskeletal Signaling
	Myristoylated PKCε inhibitor peptide（Myr-PKCε-）是一种与肉豆蔻酸偶联、具有细胞渗透性的PKCε蛋白激酶Cε亚型特异性肽抑制剂，它能够降低人脐静脉内皮细胞（HUVECs）的一氧化氮（NO）释放。
T80508	PKCη pseudosubstrate inhibitor,myristoylated	PKC	Chromatin/Epigenetic; Cytoskeletal Signaling
	Myristoylated PKCη pseudosubstrate inhibitor 是一种具有细胞渗透性的化合物，它主要应用于研究PKCη的作用机制。
T5423	PKC-theta inhibitor	PKC	Chromatin/Epigenetic; Cytoskeletal Signaling
	PKC-theta inhibitor 是一种PKC-θ抑制剂，IC50值为 12 nM。
T81450	PKCε Inhibitor Scramble Peptide
	PKCε Inhibitor Scramble Peptide为一Scramble肽，其氨基酸序列与PKCε抑制肽相同。
T80504	ɛPKC(85–92),Myristoylated	PKC	Chromatin/Epigenetic; Cytoskeletal Signaling
	PKC(85-92)，Myristoylated 是一种结合肉豆蔻酸的细胞渗透性肽，作为 PKC 激活剂，可以增强HUVECs的NO释放。
T80507	PKCθ pseudosubstrate peptide inhibitor,myristoylated	PKC	Chromatin/Epigenetic; Cytoskeletal Signaling
	Myristoylated PKCθ pseudosubstrate peptide inhibitor 是一款合成肽，专门用于研究 PKCθ 的机制。
T80070	PKCβII Peptide Inhibitor I	PKC	Chromatin/Epigenetic; Cytoskeletal Signaling
	PKCβII Peptide Inhibitor I 为一种特定的PKCβII抑制剂。在大鼠心脏缺血/再灌注损伤模型中，该化合物显著表现出心脏保护效应，并能有效预防血管内皮功能障碍。
T81449	PKC-ε translocation inhibitor peptide	PKC	Chromatin/Epigenetic; Cytoskeletal Signaling
	PKC-ε translocation inhibitor peptide，作为一种特定的PKC-ε易位抑制剂，能够特异性地调控FcγR介导的调理珠内化速率，而对FcαR运输不产生影响。
T80509	PKC 20-28,myristoylated Myristoylated protein kinase C inhibitor 20-28	PKC	Chromatin/Epigenetic; Cytoskeletal Signaling
	PKC20-28,myristoylated（Myristoylated protein kinase C inhibitor 20-28）为具细胞渗透性之PKC抑制剂，可抑制AngII所诱导之IKca电流激活，用途涵盖癌症与心血管疾病研究。
T80505	PKCα (C2-4) inhibitor peptide	PKC	Chromatin/Epigenetic; Cytoskeletal Signaling
	PKCα(C2-4) inhibitor peptide为专一性PKCα抑制剂，能够抑制α1A‐肾上腺素受体激动剂A-61603对IKr通道的影响。
T9863	PKCiota-IN-2 PKCiota-IN-49	PKC	Chromatin/Epigenetic; Cytoskeletal Signaling
	PKCiota-IN-2 (PKCiota-IN-49) 是一种有效的 PKCiota (PKC-ι) 抑制剂，IC50 为 2.8 nM。PKCiota-IN-2 还抑制 PKC-α 和 PKC-ε，IC50 分别为 71 nM 和 350 nM。
T20168	Aurothiomalate sodium 金硫丁二钠,Myocrisin,Myocrisine,Miochrysin,Sodium aurothiomalate,Myochrysine,gold sodium thiomalate	Others; PKC	Chromatin/Epigenetic; Cytoskeletal Signaling; Others
	Aurothiomalate sodium (Miochrysin) 是一种选择性的致癌 PKCι信号传导抑制剂，可抑制肿瘤细胞增殖。它是一种硫氧还蛋白还原酶 (TrxR) 抑制剂，也是一种抗风湿剂。
T72919	PKCiota-IN-1
	PKCiota-IN-1 是一种有效的 PKCiota (PKC-ι)抑制剂，IC50为 2.7 nM。PKCiota-IN-1 还抑制PKC-α和PKC-ε，IC50分别为 45 nM 和 450 nM。

化合物

PKC β pseudosubstrate acetate

Cat.No: TP1955L

Synonym: PKC β pseudosubstrate醋酸盐,Protein kinase C beta pseudosubstrate,PKC beta pseudosubstrate,PKC β pseudosubstrate acetate (172308-76-8 Free base)

Target: PKC

PKCβ inhibitor 1

Cat.No: T8376

Synonym: KUN79359

Target: Apoptosis, PKC

Cat.No: T12494

Target: PKC

PKC ζ pseudosubstrate acetate

Cat.No: TP1956L

Synonym: PKC ζ pseudosubstrate acetate (799764-07-1 free base)

Target: PKC

PKC-iota inhibitor 1

Cat.No: T8764

Target: PKC

PKCε Inhibitor Peptide acetate

Cat.No: T35827L

Synonym: PKCε Inhibitor Peptide acetate(182683-50-7 Free base)

Target: PKC

PKC-theta inhibitor hcl

Cat.No: T5817

Synonym: PKC-theta inhibitor

Target: PKC

Cat.No: T35827

Synonym: PKCε Inhibitor Peptide,Protein Kinase Cɛ Inhibitor Peptide,ɛV1-2

PKC fragment (530-558)

Cat.No: T35826

PKCζ/ι pseudosubstrate inhibitor

Cat.No: T80071

PKC β pseudosubstrate TFA

Cat.No: T75885

PKCδ Peptide Substrate

Cat.No: T76412

Cat.No: T61604

Cat.No: T71993

PKCδ Substrate TFA

Cat.No: T83754

Synonym: Protein Kinase Cδ Substrate

PKCε (85-92)

Cat.No: T80248

Target: PKC

Aurora A/PKC-IN-1

Cat.No: T62945

PKCε inhibitor peptide,myristoylated

Cat.No: T80511

Synonym: Myr‐PKCɛ-

Target: PKC

PKCη pseudosubstrate inhibitor,myristoylated

Cat.No: T80508

Target: PKC

PKC-theta inhibitor

Cat.No: T5423

Target: PKC

PKCε Inhibitor Scramble Peptide

Cat.No: T81450

ɛPKC(85–92),Myristoylated

Cat.No: T80504

Target: PKC

PKCθ pseudosubstrate peptide inhibitor,myristoylated

Cat.No: T80507

Target: PKC

PKCβII Peptide Inhibitor I

Cat.No: T80070

Target: PKC

PKC-ε translocation inhibitor peptide

Cat.No: T81449

Target: PKC

PKC 20-28,myristoylated

Cat.No: T80509

Synonym: Myristoylated protein kinase C inhibitor 20-28

Target: PKC

PKCα (C2-4) inhibitor peptide

Cat.No: T80505

Target: PKC

Cat.No: T9863

Synonym: PKCiota-IN-49

Target: PKC

Aurothiomalate sodium

Cat.No: T20168

Synonym: 金硫丁二钠,Myocrisin,Myocrisine,Miochrysin,Sodium aurothiomalate,Myochrysine,gold sodium thiomalate

Target: Others, PKC

Cat.No: T72919

Species：

Expression System：

Tag：

Cat. No.	Product Name	Species	Expression System
TMPY-04455	PKC iota Protein, Human, Recombinant (GST) PKCI,nPKC-iota,protein kinase C, ι	Human	Baculovirus Insect Cells
	Protein kinase C iota type, also known as Atypical protein kinase C-lambda/iota, aPKC-lambda/iota and PRKCI, is a cytoplasm, membrane and nucleus protein which belongs to the protein kinase superfamily, AGC Ser/Thr protein kinase family and PKC subfamily. PRKCI contains one AGC-kinase C-terminal domain, one OPR domain, one phorbol-ester/DAG-type zinc finger and one protein kinase domain. PRKCI is predominantly expressed in lung and brain, but also expressed at lower levels in many tissues includ...
TMPY-04456	PKC nu Protein, Human, Recombinant (GST) PRKCN,nPKC-NU,PKC-NU,PKD3,EPK2,protein kin...	Human	Baculovirus Insect Cells
	Serine/threonine-protein kinase D3, also known as Protein kinase C nu type, Protein kinase EPK2, PRKD3, EPK2 and PRKCN, is a cytoplasm and membrane protein that belongs to the protein kinase superfamily, CAMK Ser/Thr protein kinase family and PKD subfamily. PRKD3 / PRKCN contains one PH domain, two phorbol-ester/DAG-type zinc fingers and one protein kinase domain. Protein kinase C (PKC) is a family of serine- and threonine-specific protein kinases that can be activated by calcium and the second ...

重组蛋白

PKC iota Protein, Human, Recombinant (GST)

Cat.No: TMPY-04455

Species: Human

Expression System: Baculovirus Insect Cells

PKC nu Protein, Human, Recombinant (GST)

Cat.No: TMPY-04456

Species: Human

Expression System: Baculovirus Insect Cells

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